5U9D | pdb_00005u9d

Discovery of a potent BTK inhibitor with a novel binding mode using parallel selections with a DNA-encoded chemical library

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CHAIN
A
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform - Homo sapiens
 Explore Sequence Annotations in 3D
0100200300400500600700800900
CHAIN A
UNIPROT P48736
SECONDARY STRUCTURE
UNMODELED
PLANE OUTLIERS
EDS ATOMS
OCC WT AVG B
AVERAGE OCCUPANCY
ATOMIC CLASHES
ANGLE OUTLIERS
RSRZ
RSR
RSCC
CIS-PEPTIDE
BINDING SITE 1JV
BURIED RESIDUES
ARTIFACT
HYDROPATHY
DISORDER
DISORDERED BINDING
PFAM
CATH
SCOP
ECOD
MOLECULE PROCESSING
GENOME VARIANT
MODIFIED RESIDUE
MUTAGENESIS
CONFLICT
DOMAIN
REGION