2FWY | pdb_00002fwy

Structure of human Hsp90-alpha bound to the potent water soluble inhibitor PU-H64

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RCSB PDB Mol* Viewer 2.11.4 [4/4/2025, 6:48:47 PM]
Sequence of
     ​M​​G​​S​​S​​H​​H​​H​​H​​H​​H​     ​S​​S​​G​​L​​V​​P​​R​​G​​S​​H​     ​M​​P​​E​​E​​T​​Q​​T​​Q​​D​​Q​     ​P​​M​​E​​E​​E​​E​​V​​E​​T​​F​21   ​A​​F​​Q​​A​​E​​I​​A​​Q​​L​​M​31   ​S​​L​​I​​I​​N​​T​​F​​Y​​S​​N​41   ​K​​E​​I​​F​​L​​R​​E​​L​​I​​S​51   ​N​​S​​S​​D​​A​​L​​D​​K​​I​​R​61   ​Y​​E​​S​​L​​T​​D​​P​​S​​K​​L​71   ​D​​S​​G​​K​​E​​L​​H​​I​​N​​L​81   ​I​​P​​N​​K​​Q​​D​​R​​T​​L​​T​91   ​I​​V​​D​​T​​G​​I​​G​​M​​T​​K​101  ​A​​D​​L​​I​​N​​N​​L​​G​​T​​I​111  ​A​​K​​S​​G​​T​​K​​A​​F​​M​​E​121  ​A​​L​​Q​​A​​G​​A​​D​​I​​S​​M​131  ​I​​G​​Q​​F​​G​​V​​G​​F​​Y​​S​141  ​A​​Y​​L​​V​​A​​E​​K​​V​​T​​V​151  ​I​​T​​K​​H​​N​​D​​D​​E​​Q​​Y​161  ​A​​W​​E​​S​​S​​A​​G​​G​​S​​F​171  ​T​​V​​R​​T​​D​​T​​G​​E​​P​​M​181  ​G​​R​​G​​T​​K​​V​​I​​L​​H​​L​191  ​K​​E​​D​​Q​​T​​E​​Y​​L​​E​​E​201  ​R​​R​​I​​K​​E​​I​​V​​K​​K​​H​211  ​S​​Q​​F​​I​​G​​Y​​P​​I​​T​​L​221  ​F​​V​​E​​K​​E​​R​​D​​K​​E​​V​     ​S​​D​​D​​E​​A​​E​
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